4-[[(7R)-8-環戊基-7-乙基-5,6,7,8-四氫-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺抑制劑BI2536 is an effective Plk1 inhibitor (IC50: 0.83 nM). It has 4- and 11-fold greater selectivity than Plk2 and Plk3.
產品名稱: | 4-[[(7R)-8-環戊基-7-乙基-5,6,7,8-四氫-5-甲基-6-氧代-2-喋啶基]氨基]-3-甲氧基-N-(1-甲基-4-哌啶基)苯甲酰胺 | ||
英文名: | BI 2536 | ||
CAS NO.: | 755038-02-9 | ||
分子式: | C28H39N7O3 | ||
分子量: | 521.654365777969 | ||
產品品牌: | targetmol | ||
產品規格: | 2mg |