ML221抑制劑ML221 is a potent?apelin /APJ?functional antagonist, inhibiting apelin-13-mediated activation of APJ, with?IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and?EC80?of 10 nM in both assays.
產品名稱: | ML221 | ||
英文名: | ML221 | ||
CAS NO.: | 877636-42-5 | ||
分子式: | C17H11N3O6S | ||
分子量: | 385.350742578506 | ||
產品品牌: | targetmol | ||
產品規格: | 1mg |